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In emergencies, such as hyperglycemic coma, it can be given intravenously (mostly by infusion because i. v. injections have too brief an action; plasma t1/2 ~ 9 min). With the usual subcutaneous application, the effect is evident within 15 to 20 min, reaches a peak after approx. 3 h, and lasts for approx. 6 h. Lispro insulin has a faster onset and slightly shorter duration of action.
Oral anticoagulants. Structurally related to vitamin K, 4-hydroxycoumarins act as “false” vitamin K and prevent regeneration of reduced (active) vitamin K from vitamin K epoxide, hence the synthesis of vitamin K-dependent clotting factors. Coumarins are well absorbed after oral administration. Their duration of action varies considerably. |
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